SCHEMBL23846503

SCHEMBL23846503

COc1ccc(N)cc1S(=O)(=O)Nc1ccc(C)cc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.71
HTT P42858 1/20 0.71
LMNA P02545 3/20 0.67
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
GAA P10253 2/20 0.66
HDAC1 Q13547 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
RECQL P46063 1/20 0.63
HPGD P15428 3/20 0.62
ALDH1A1 P00352 3/20 0.56
THRB P10828 1/20 0.56
NPSR1 Q6W5P4 2/20 0.55
ALPL P05186 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2241241 0.89 SMN1; SMN2 (0.59) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL25754817 0.87 NPSR1 (0.62) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL17980891 0.87 MAPT (0.60) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL23846500 0.87 LMNA (0.73) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL23847019 0.87 MEN1 (0.61) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL23847027 0.86 MEN1 (0.59) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL25754779 0.85 MEN1 (0.80) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL23846529 0.85 ALPL (0.60) SMN1; SMN2HTTLMNAMEN1KMT2A
SCHEMBL23833758 0.84 RECQL (0.73) SMN1; SMN2LMNAGAARECQLALDH1A1
SCHEMBL23833737 0.84 MEN1 (0.63) SMN1; SMN2HTTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
WO-2021188880-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 SMN1; SMN2 405/4885HTT 69/4885LMNA 3435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.