SCHEMBL23886102

SCHEMBL23886102

Cc1cccc2nc(Cc3ccccc3)c(Cl)nc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PTPN1 P18031 1/20 0.40
MAOA P21397 2/20 0.40
HRH4 Q9H3N8 2/20 0.40
MAOB P27338 1/20 0.40
HRH1 P35367 1/20 0.40
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
RXFP1 Q9HBX9 2/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30177343 1.00 DRD4 (0.46) DRD4DRD3L3MBTL1KDM4EALDH1A1
SCHEMBL23885969 0.94 L3MBTL1 (0.43) DRD4DRD3L3MBTL1KDM4EALDH1A1
SCHEMBL3611417 0.80 TDP1 (0.54) KDM4EALDH1A1GAAHPGDHTT
SCHEMBL2423180 0.76 TDP1 (0.52) DRD4DRD3L3MBTL1KDM4EALDH1A1
SCHEMBL31399980 0.76 TDP1 (0.52) DRD4DRD3L3MBTL1KDM4EALDH1A1
SCHEMBL14764415 0.73 MAPT (0.44) DRD4DRD3L3MBTL1ALDH1A1GAA
SCHEMBL6311606 0.72 HRH4 (0.45) L3MBTL1KDM4EALDH1A1GAAHPGD
SCHEMBL28118305 0.70 GAA (0.56) KDM4EALDH1A1GAAHPGDHTT
SCHEMBL14842553 0.70 KDM4E (0.62) L3MBTL1KDM4EALDH1A1GAAHPGD
SCHEMBL20475325 0.70 RAB9A (0.53) ALDH1A1GAAMAPTMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12428403-B2 N-(heterocyclyl and heterocyclylalkyl)-3-benzylpyridin-2-amine derivatives as SSTR4 agonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2025-09-30 US disclosed
CN-115485273-B N- (heterocyclyl and heterocyclylalkyl) -3-benzyl pyridin-2-amine derivatives as SSTR4 agonists 武田药品工业株式会社 2024-08-13 CN disclosed
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-06-22 US disclosed
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-06-22 US disclosed
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-06-22 US disclosed
EP-4126849-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS Takeda Pharmaceutical Company Limited (JP) 2023-02-08 EP disclosed
CN-115485273-A N- (heterocyclyl and heterocyclylalkyl) -3-benzylpyridin-2-amine derivatives as SSTR4 agonists 武田药品工业株式会社 2022-12-16 CN disclosed
WO-2021202775-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-10-07 WO disclosed
WO-2021202775-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12428403-B2 N-(heterocyclyl and heterocyclylalkyl)-3-benzylpyridin-2-amine derivatives as SSTR4 agonists SSTR4, SSTR3, SSTR1 DRD4 415/4885DRD3 549/4885L3MBTL1 4683/4885
US-20230192659-A1 N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS SSTR4, SSTR3, SSTR1 DRD4 415/4885DRD3 549/4885L3MBTL1 4683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.