SCHEMBL2389201

SCHEMBL2389201

O=C(Cc1cccnc1)Nc1ccc2c(c1)Oc1ccc(NC(=O)Cc3cccnc3)cc1O2

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.62
PSMB8 P28062 2/20 0.57
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
ESR1 P03372 1/20 0.54
POLB P06746 1/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
ROCK1 Q13464 1/20 0.52
PDE3B Q13370 1/20 0.50
EPHX2 P34913 1/20 0.48
HTR1A P08908 2/20 0.48
DRD2 P14416 2/20 0.48
MAPK8 P45983 1/20 0.48
NAPRT Q6XQN6 1/20 0.48
GLS O94925 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2388252 0.83 RAB9A (0.64) KDM4EUSP2ALDH1A1EPHX2NPC1
SCHEMBL362394 0.80 ALDH1A1 (0.66) PSMB8ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL13766306 0.77 SMN1; SMN2 (0.58) ROCK2PSMB8POLBHPGDCYP1A2
SCHEMBL17783810 0.77 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL14073604 0.77 ROCK2 (0.60) ROCK2PSMB8ALDH1A1CYP1A2CYP3A4
SCHEMBL14073866 0.77 ROCK2 (0.63) ROCK2PSMB8CYP1A2CYP3A4CYP2C9
SCHEMBL10759415 0.77 PSMB8 (0.55) ROCK2PSMB8KDM4EUSP2ALDH1A1
SCHEMBL25810554 0.77 MEN1 (0.57) ROCK2PSMB8ALDH1A1HPGDCYP1A2
SCHEMBL25380516 0.76 CFD (0.62) PSMB8KDM4EUSP2ALDH1A1ESR1
SCHEMBL30510132 0.76 CFD (0.62) PSMB8KDM4EUSP2ALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012606-B2 Heterocyclic compound and organic electroluminescent device using the same NIPPON STEEL CHEMICAL CO., LTD. (JP) 2011-09-06 US disclosed
US-20090153031-A1 Heterocyclic compound and organic electroluminescent device using the same NIPPON STEEL CHEMICAL CO., LTD (JP) 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090153031-A1 Heterocyclic compound and organic electroluminescent device using the same ORC3, NAP1L4, NR4A2 ROCK2 3060/4885PSMB8 2545/4885KDM4E 1619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.