SCHEMBL23901095

SCHEMBL23901095

Nc1n[nH]c2ccc(C(COCc3ccccc3)c3cc(F)cc(F)c3)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.41
CDC7 O00311 8/20 0.41
CDK2 P24941 7/20 0.41
ROCK2 O75116 7/20 0.41
PRKACA P17612 6/20 0.41
GSK3B P49841 6/20 0.41
AURKB Q96GD4 6/20 0.41
JAK3 P52333 6/20 0.41
MAP4K4 O95819 5/20 0.41
CLK4 Q9HAZ1 5/20 0.41
MKNK2 Q9HBH9 5/20 0.41
MAPK13 O15264 5/20 0.41
DAPK3 O43293 5/20 0.41
PRKCG P05129 5/20 0.41
CDK1 P06493 5/20 0.41
MARK3 P27448 5/20 0.41
GSK3A P49840 5/20 0.41
MAPK12 P53778 5/20 0.41
CSNK2A1 P68400 5/20 0.41
CDK5 Q00535 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23901216 0.82 MAPK1 (0.43) JAK2CDC7CDK2ROCK2PRKACA
SCHEMBL23901318 0.80 JAK2 (0.43) JAK2CDC7CDK2ROCK2PRKACA
SCHEMBL23901101 0.72 TACR1 (0.39) TACR1GAA
SCHEMBL3509883 0.72 JAK2 (0.45) JAK2CDC7CDK2ROCK2PRKACA
SCHEMBL28999529 0.70 TACR1 (0.37) TACR1
SCHEMBL28999399 0.70 JAK2 (0.43) JAK2CDC7CDK2ROCK2PRKACA
SCHEMBL627903 0.69 TTK (0.59) JAK2NTRK1KDM4EGAA
SCHEMBL30451203 0.69 NTRK1 (0.66) JAK2AURKBNTRK1AURKAPDPK1
SCHEMBL3510229 0.69 NTRK1 (0.66) JAK2AURKBNTRK1AURKAPDPK1
SCHEMBL3512392 0.68 JAK2 (0.58) JAK2CDC7CDK2ROCK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-B Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2025-04-01 CN disclosed
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed