SCHEMBL28999529

SCHEMBL28999529

N#Cc1cc(C(COCc2ccccc2)c2cc(F)cc(F)c2)ccc1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.37
MAOB P27338 1/20 0.37
CA1 P00915 4/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
CTSL P07711 1/20 0.34
TSHR P16473 1/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23901101 0.81 TACR1 (0.39) TACR1CA1CA2CA7CA9
SCHEMBL23901224 0.81 PTGDR2 (0.34)
SCHEMBL31391641 0.81 PTGDR2 (0.34)
SCHEMBL23901317 0.77 PTGDR2 (0.37)
SCHEMBL23901319 0.76 ADRB2 (0.40)
SCHEMBL31391663 0.70 TACR1 (0.39) TACR1CA1CA2CA7CA9
SCHEMBL23901095 0.70 JAK2 (0.41) TACR1
SCHEMBL4753464 0.69 MAOB (0.74) MAOB
SCHEMBL22469496 0.69 TSHR (0.47) MAOBCTSBCTSLTSHRBACE1
SCHEMBL3511297 0.68 ADRB2 (0.37) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed