SCHEMBL23901101

SCHEMBL23901101

Fc1cc(F)cc(C(COCc2ccccc2)c2ccc(F)c(Br)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.39
CA1 P00915 4/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
TSHR P16473 1/20 0.36
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34
MEN1 O00255 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28999529 0.81 TACR1 (0.37) TACR1CA1CA2CA7CA9
SCHEMBL23901223 0.79 SLC6A2 (0.33) IDO1TDO2
SCHEMBL31391663 0.78 TACR1 (0.39) TACR1CA1CA2CA7CA9
SCHEMBL23901091 0.74 ADRB2 (0.35) IDO1TDO2
SCHEMBL11139289 0.74 TSHR (0.54) TSHRIDO1TDO2
SCHEMBL23901095 0.72 JAK2 (0.41) TACR1GAA
SCHEMBL31391702 0.71 DPP4 (0.31)
SCHEMBL28999511 0.71 DPP4 (0.31)
SCHEMBL29870987 0.67 MAOB (0.43) TSHR
SCHEMBL26428048 0.67 MAOB (0.43) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed