SCHEMBL23905655

SCHEMBL23905655

COc1cc(C(=O)NCC(c2cc3c(c(-c4ccc(C(F)(F)F)cc4)n2)OCC3(CF)CF)C2CC2)cc2cc(Cl)nnc12

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
MDM2 Q00987 1/20 0.31
CTSA P10619 1/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
MAPT P10636 1/20 0.30
MTTP P55157 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905976 0.93 MAPT (0.32) ADRA1DADRA1AADRA1BROCK2ROCK1
SCHEMBL23905652 0.84 ADRA1D (0.34) ADRA1DADRA1AADRA1BMAPT
SCHEMBL23905991 0.84 ROCK2 (0.32) ROCK2ROCK1MAPTMTTP
SCHEMBL23905665 0.83 MAPT (0.33) ROCK2ROCK1MAPT
SCHEMBL23905980 0.83 ADRA1D (0.33) ADRA1DADRA1AADRA1BROCK2ROCK1
SCHEMBL23905959 0.83 MAPT (0.34) ADRA1DADRA1AADRA1BROCK2ROCK1
SCHEMBL23905961 0.81 MAPT (0.32) ADRA1DADRA1AADRA1BCTSAROCK2
SCHEMBL23904705 0.80
SCHEMBL23905824 0.79
SCHEMBL23905985 0.77 PTGFR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198981-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF Janssen Biopharma, Inc. (US) 2021-10-07 WO disclosed