SCHEMBL23905955

SCHEMBL23905955

CC(C)c1c(OCc2cccc(C#N)c2)ccc2c1OCCC2=O

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.60
MAOB P27338 8/20 0.49
MAOA P21397 1/20 0.49
MRGPRX4 Q96LA9 4/20 0.43
HTR6 P50406 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SLC6A4 P31645 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905971 0.87 GRM5 (0.63) GRM5MAOBMAOAMRGPRX4HTR6
SCHEMBL23882634 0.79 MAOB (0.42) GRM5MAOBMRGPRX4NPC1ALDH1A1
SCHEMBL32675527 0.79 MAOB (0.42) GRM5MAOBMRGPRX4NPC1ALDH1A1
SCHEMBL23905943 0.78 GRM5 (0.41) GRM5MAOBMRGPRX4NPC1ALDH1A1
SCHEMBL23882644 0.77 MAOB (0.47) GRM5MAOBMAOANPC1ALDH1A1
SCHEMBL23906321 0.77 GRM5 (0.39) GRM5MAOBMAOA
SCHEMBL23906005 0.76 RXRA (0.46) GRM5MAOBMRGPRX4NPC1ALDH1A1
SCHEMBL23905950 0.75 GRM5 (0.38) GRM5MAOBMAOA
SCHEMBL30251244 0.75 GRM5 (0.38) GRM5MAOBMAOA
SCHEMBL30251163 0.75 GRM5 (0.38) GRM5MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021198283-A1 INHIBITORS OF ANTIGEN PRESENTATION BY HLA-DR JANSSEN PHARMACEUTICA NV (BE) 2021-10-07 WO disclosed