SCHEMBL23912554

SCHEMBL23912554

CCc1cc(OC)c(O)nn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.36
HMGCR P04035 2/20 0.36
MAPT P10636 2/20 0.34
CYP3A4 P08684 1/20 0.34
SMPD3 Q9NY59 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 3/20 0.33
GAA P10253 2/20 0.33
POLB P06746 1/20 0.33
ALOX5 P09917 4/20 0.33
PTGS1 P23219 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
MAOB P27338 1/20 0.32
KDM4E B2RXH2 2/20 0.32
NFKB1 P19838 1/20 0.32
PGK1 P00558 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24226822 0.73 TAAR1 (0.36) PTGS2SMPD3SMN1; SMN2ALDH1A1TAAR1
SCHEMBL13082756 0.73 PTGS2 (0.34) PTGS2CYP3A4SMN1; SMN2ALDH1A1GAA
SCHEMBL30646151 0.72 KMT2A (0.41) HMGCRSMN1; SMN2
SCHEMBL22042471 0.71 ALDH1A1 (0.40) PTGS2MAPTCYP3A4SMN1; SMN2ALDH1A1
SCHEMBL23912350 0.68 SMN1; SMN2 (0.38) MAPTSMN1; SMN2ALDH1A1KDM4EPDE4A
SCHEMBL12202933 0.67 P2RX3 (0.41) PTGS2HMGCRMAPTCYP3A4SMN1; SMN2
SCHEMBL118146 0.66 CYP3A4 (0.44) PTGS2MAPTCYP3A4SMPD3ALDH1A1
SCHEMBL24920246 0.64 PDE4A (0.32) MAPTCYP3A4SMN1; SMN2POLBKDM4E
SCHEMBL13952464 0.64 PTGS2 (0.36) PTGS2ALDH1A1TAAR1
SCHEMBL72546 0.64 PDE4A (0.39) MAPTCYP3A4ALDH1A1TAAR1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892278-B1 CYCLOALKANE-1,3-DIAMINE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2024-02-28 EP disclosed
EP-3892278-A1 CYCLOALKANE-1,3-DIAMINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-10-13 EP disclosed