SCHEMBL23912778

SCHEMBL23912778

CNc1cc(B2OC(C)(C)C(C)(C)O2)c(C)cn1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.38
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
LIPE Q05469 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12456123 0.81 UHRF1 (0.35) CYP1A2MAPK1
SCHEMBL29781537 0.81 UHRF1 (0.35) CYP1A2MAPK1
SCHEMBL626900 0.80 L3MBTL1 (0.44) CYP1A2LIPE
SCHEMBL30508802 0.78 LPL (0.35) LIPEMAPK1
SCHEMBL15342466 0.78 EGFR (0.31) MAPK1
SCHEMBL1192473 0.78 LPL (0.35) LIPEMAPK1
SCHEMBL15051210 0.76 ABL1 (0.46)
SCHEMBL29652860 0.75 NNMT (0.37) NNMTLIPE
SCHEMBL20519939 0.75 NNMT (0.37) NNMTLIPE
SCHEMBL30508803 0.75 LPL (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3094325-B1 HETEROARYLS AND USES THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2021-10-13 EP disclosed