SCHEMBL23917013

SCHEMBL23917013

CS(=O)(=O)c1nc(OCC(=O)NC23CC4CC(CC(C4)C2)C3)c(F)c(N2CCOCC2)n1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CNR2 P34972 4/20 0.41
EPHX2 P34913 5/20 0.38
ALDH1A1 P00352 6/20 0.37
LMNA P02545 2/20 0.37
CNR1 P21554 1/20 0.36
TSHR P16473 2/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23907982 0.85 CNR2 (0.41) MEN1KMT2ACNR2EPHX2ALDH1A1
SCHEMBL23884289 0.82 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL30165249 0.82 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL23884199 0.77 MEN1 (0.42) MEN1KMT2ACNR2EPHX2ALDH1A1
SCHEMBL23907983 0.72 ALDH1A1 (0.38) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL23884309 0.71 LMNA (0.48) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL23900379 0.70 MEN1 (0.43) MEN1KMT2ACNR2EPHX2ALDH1A1
SCHEMBL23900313 0.70 ALDH1A1 (0.46) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL23907992 0.69 EPHX2 (0.46) KMT2AEPHX2ALDH1A1LMNATSHR
SCHEMBL23884322 0.67 ALDH1A1 (0.43) MEN1KMT2AALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230120566-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses OREGON HEALTH AND SCIENCE UNIVERSITY 2023-04-20 US disclosed
US-11566019-B2 2-pyrimidone analogs as potent antiviral agents against alphaviruses SOUTHERN RESEARCH INSTITUTE (US) 2023-01-31 US disclosed
US-20220177452-A9 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-06-09 US disclosed
US-20210317106-A1 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses SOUTHERN RES INST (US) 2021-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317106-A1 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS MEN1 4254/4885KMT2A 2117/4885CNR2 4380/4885
US-11566019-B2 2-pyrimidone analogs as potent antiviral agents against alphaviruses EIF2AK2, ZC3HAV1, MAVS MEN1 4254/4885KMT2A 2117/4885CNR2 4380/4885
US-20220177452-A9 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS MEN1 4254/4885KMT2A 2117/4885CNR2 4380/4885
US-20230120566-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS MEN1 4347/4885KMT2A 2305/4885CNR2 4247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.