SCHEMBL23922755

SCHEMBL23922755

O=Cc1ccc(N2CCN(Cc3ccncc3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.63
TRIM24 O15164 1/20 0.51
TRIM33 Q9UPN9 1/20 0.51
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
DRD4 P21917 4/20 0.49
CASP1 P29466 1/20 0.47
CASP4 P49662 1/20 0.47
CASP5 P51878 1/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
MAPT P10636 1/20 0.46
LSS P48449 1/20 0.44
KHK P50053 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4392263 0.85 DRD4 (0.70) TRIM24TRIM33ALDH1A1KDM4ESMN1; SMN2
SCHEMBL7958672 0.84 TRIM24 (0.66) TRIM24TRIM33ALDH1A1KDM4ESMN1; SMN2
SCHEMBL28710553 0.83 HDAC3 (0.57) POLBALDH1A1KDM4ESMN1; SMN2DRD4
SCHEMBL27371894 0.81 DRD4 (0.71) POLBALDH1A1KDM4EDRD4DRD2
SCHEMBL1509470 0.80 POLB (0.63) POLBALDH1A1KDM4ESMN1; SMN2DRD4
SCHEMBL1669246 0.80 DRD4 (0.77) POLBALDH1A1KDM4EDRD4DRD2
SCHEMBL27990811 0.79 HRH3 (0.52) POLBTRIM24TRIM33ALDH1A1KDM4E
SCHEMBL4579770 0.78 POLB (0.61) POLBALDH1A1KDM4ESMN1; SMN2DRD4
SCHEMBL28710385 0.78 ALDH1A1 (0.47) POLBTRIM24TRIM33ALDH1A1KDM4E
SCHEMBL27373181 0.78 POLB (0.60) POLBALDH1A1KDM4EDRD4CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481824-B1 2-PHENYLIMIDAZO[4,5-B]PYRIDIN-7-AMINE DERIVATES USEFUL AS INHIBITORS OF MAMMALIAN TYROSINE KINASE ROR1 ACTIVITY KANCERA AB (SE) 2021-10-20 EP disclosed
CN-109563092-B 2-phenylimidazo [4,5-B ] pyridin-7-amine derivatives useful as inhibitors of the activity of the mammalian tyrosine kinase ROR1 坎塞拉有限公司 2021-09-14 CN disclosed