SCHEMBL23928141

SCHEMBL23928141

CN(C)C1CCN(CCOc2ccc(CCNC(=O)OCc3ccccc3)cc2)C1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
LTA4H P09960 14/20 0.51
MC4R P32245 1/20 0.50
KDM4E B2RXH2 1/20 0.49
HRH3 Q9Y5N1 2/20 0.48
CCR5 P51681 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26964861 1.00 MAPT (0.52) MAPTL3MBTL1LTA4HMC4RKDM4E
SCHEMBL26964857 1.00 MAPT (0.52) MAPTL3MBTL1LTA4HMC4RKDM4E
SCHEMBL23928187 0.87 HRH3 (0.54) LTA4HMC4RHRH3
SCHEMBL23291139 0.87 HRH3 (0.54) LTA4HMC4RHRH3
SCHEMBL23291207 0.85 MAPT (0.61) MAPTL3MBTL1LTA4HMC4RKDM4E
SCHEMBL23291140 0.83 HTT (0.61) MAPTL3MBTL1LTA4HKDM4EHRH3
SCHEMBL30011423 0.80 KEAP1 (0.52) L3MBTL1HRH3CCR5
SCHEMBL23291310 0.79 MC4R (0.48) MAPTLTA4HMC4RKDM4EHRH3
SCHEMBL23291169 0.78 ITGB3 (0.64) MAPTL3MBTL1LTA4HKDM4EHRH3
SCHEMBL22482290 0.77 LMNA (0.52) MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3814356-B1 TRIAZOLOTRIAZINE DERIVATIVES AS A2A RECEPTOR ANTAGONISTS ZHEJIANG VIMGREEN PHARMACEUTICALS LTD (CN) 2026-03-11 EP disclosed
US-11845751-B2 Triazolotriazine derivatives as A2A receptor antagonists ZHEJIANG VIMGREEN PHARMACEUTICALS, LTD. (CN) 2023-12-19 US disclosed
CN-111051309-B Triazolotriazine derivatives useful as A2A receptor antagonists 浙江春禾医药科技有限公司 2023-05-26 CN disclosed
US-20210332055-A1 TRIAZOLOTRIAZINE DERIVATIVES AS A2A RECEPTOR ANTAGONISTS ZHEJIANG VIMGREEN PHARMACEUTICALS, LTD. (CN) 2021-10-28 US disclosed
CN-111051309-A Triazolotriazine derivatives useful as A2A receptor antagonists 浙江春禾医药科技有限公司 2020-04-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11845751-B2 Triazolotriazine derivatives as A2A receptor antagonists ADORA2A, ADORA1, ADORA3 MAPT 3868/4885L3MBTL1 4623/4885LTA4H 1029/4885
US-20210332055-A1 TRIAZOLOTRIAZINE DERIVATIVES AS A2A RECEPTOR ANTAGONISTS ADORA2A, ADORA1, ADORA3 MAPT 3868/4885L3MBTL1 4623/4885LTA4H 1029/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.