SCHEMBL2392990

SCHEMBL2392990

Fc1ccc(NC(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
CFTR P13569 1/20 0.48
GOPC Q9HD26 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 3/20 0.47
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TEAD4 Q15561 1/20 0.43
CA12 O43570 1/20 0.42
MMP2 P08253 1/20 0.42
RCE1 Q9Y256 3/20 0.42
KLK7 P49862 1/20 0.41
RAB9A P51151 2/20 0.41
MTOR P42345 1/20 0.41
GRM7 Q14831 1/20 0.41
NPC1 O15118 1/20 0.41
NOX1 Q9Y5S8 1/20 0.41
KCNH3 Q9ULD8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361907 0.84 CFTR (0.63) KMT2ACFTRGOPCKDM4EMEN1
SCHEMBL7348000 0.79 ALDH1A1 (0.62) KMT2AKDM4EMEN1NPC1KCNH3
SCHEMBL15003944 0.79 ALDH1A1 (0.62) KMT2AKDM4EMEN1NPC1KCNH3
SCHEMBL28359204 0.78 KMT2A (0.77) KMT2ACFTRGOPCMEN1MAPT
SCHEMBL27874471 0.78 KMT2A (0.53) KMT2ACFTRGOPCKDM4EMEN1
SCHEMBL29665053 0.78 MAPT (0.52) KMT2ACFTRGOPCKDM4EMEN1
SCHEMBL28707659 0.78 KMT2A (0.51) KMT2ACFTRGOPCMEN1MAPT
SCHEMBL5512074 0.78 MAPT (0.52) KMT2ACFTRGOPCMEN1MAPT
SCHEMBL28428339 0.78 RAB9A (0.46) KMT2ACFTRGOPCKDM4EMEN1
SCHEMBL28407865 0.78 KMT2A (0.51) KMT2ACFTRGOPCMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116496211-A Large-steric-hindrance pyridine amide, nickel complex, preparation method and application thereof in olefin polymerization 安徽大学 2023-07-28 CN disclosed
CN-111205334-A High-activity complex for catalyzing ethylene polymerization and preparation method thereof 卢静 2020-05-29 CN disclosed
US-8026263-B2 Methods for inhibiting neoproliferative changes in blood vessel walls THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-09-27 US disclosed
US-20090048270-A1 Compounds, Methods And Devices for Inhibiting Neoproliferative Changes in Blood Vessel Walls NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2009-02-19 US disclosed
US-20070293554-A1 Non-peptide inhibition of T-lymphocyte activation and therapies related thereto THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2007-12-20 US disclosed
US-7235577-B1 Non-peptide inhibition of T-lymphocyte activation and therapies related thereto THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-06-26 US disclosed
US-6803375-B1 IMMUNOMODULATION IN A MAMMALIAN PATIENT WITHOUT CAUSING SUBSTANTIAL INHIBITION OF CYTOCHROME P-450 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2004-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048270-A1 Compounds, Methods And Devices for Inhibiting Neoproliferative Changes in Blood Vessel Walls PGF, VEGFA, MKI67 KMT2A 1774/4885CFTR 2376/4885GOPC 3889/4885
US-20070293554-A1 Non-peptide inhibition of T-lymphocyte activation and therapies related thereto NFATC1, ORAI1, KCNMA1 KMT2A 2461/4885CFTR 1267/4885GOPC 2587/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.