SCHEMBL23937765

SCHEMBL23937765

CCn1cc(C(N)=O)c2ccsc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
PTK2 Q05397 1/20 0.37
NR4A2 P43354 1/20 0.36
MAP2K2 P36507 1/20 0.36
MAP2K1 Q02750 1/20 0.36
BRD4 O60885 1/20 0.35
CNR1 P21554 1/20 0.35
FABP4 P15090 1/20 0.34
ICMT O60725 1/20 0.34
MAPK8 P45983 2/20 0.34
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BRCA1 P38398 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20673875 0.82 LMNA (0.43) ALDH1A1KMT2AMEN1MAPK1NR4A2
SCHEMBL11557695 0.79 LMNA (0.52) ALDH1A1KMT2AMEN1BRD4HSD17B10
SCHEMBL21958623 0.78 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL20673904 0.75 MAP2K2 (0.41) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL28070206 0.71 NR4A2 (0.68) ALDH1A1KMT2ANR4A2CNR1BRCA1
SCHEMBL11664740 0.68 LMNA (0.44) ALDH1A1KMT2AMEN1HSD17B10KDM4E
SCHEMBL28131233 0.68 ICMT (0.55) ALDH1A1KMT2AMAPTNR4A2MAP2K2
SCHEMBL10193361 0.68 CNR1 (0.46) ALDH1A1KMT2AMEN1NR4A2MAP2K2
SCHEMBL21958624 0.67 BRD4 (0.38) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL8513279 0.67 CNR1 (0.51) ALDH1A1CNR1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed