SCHEMBL23937904

SCHEMBL23937904

On1cc(C(F)(F)F)c2c1CCCCC2

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FABP4 P15090 3/20 0.34
FABP3 P05413 1/20 0.34
HTT P42858 1/20 0.33
GAA P10253 2/20 0.33
GRIA2 P42262 4/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
CA2 P00918 1/20 0.31
CYP2C19 P33261 1/20 0.31
CYP2D6 P10635 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20631118 0.94 CA2 (0.32) LMNAALDH1A1TSHRNPSR1KDM4E
SCHEMBL20631714 0.79 GRM2 (0.32)
SCHEMBL23937908 0.72 ALOX5 (0.35) KDM4E
SCHEMBL23937896 0.71 HTR2A (0.33) LMNAALDH1A1TSHRKDM4EHPGD
SCHEMBL23937907 0.70 ALOX5 (0.33) ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL23937917 0.68 HSD17B10 (0.35) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL23937926 0.67
SCHEMBL23937643 0.66 KDM4E (0.34) LMNAALDH1A1NPSR1KDM4EHTT
SCHEMBL23937899 0.65 HSD17B10 (0.33) ALDH1A1KDM4EHSD17B10CYP2C9
SCHEMBL23937911 0.64 POLB (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed