SCHEMBL23950203

SCHEMBL23950203

CCc1nn(CC)c(=O)c2ccnn12

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.39
BRD9 Q9H8M2 1/20 0.35
TBXAS1 P24557 1/20 0.35
TP53 P04637 2/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 2/20 0.34
ADORA2A P29274 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
NLRP3 Q96P20 1/20 0.34
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23950198 0.84 ALOX15 (0.47) PIK3CATP53POLBMAPTNLRP3
SCHEMBL23950524 0.79 KDM4E (0.47) POLB
SCHEMBL23950616 0.75 NLRP3 (0.50) TP53POLBMAPTNLRP3
SCHEMBL23950196 0.75 TP53 (0.56) TP53MAPTNLRP3NPC1
SCHEMBL23950623 0.73 TP53 (0.52) TP53POLBNLRP3NPC1
SCHEMBL23950622 0.70 POLB (0.60) TP53POLBMAPT
SCHEMBL23925544 0.70 PDE4B (0.34) PIK3CABRD9
SCHEMBL4194913 0.69 PIK3CA (0.36) PIK3CAPOLB
SCHEMBL15185707 0.67 KMT2A (0.38) TBXAS1MAPTNPC1
SCHEMBL14084736 0.63 RAB9A (0.42) POLBMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021209552-A1 PYRAZOLO[1,5-D][1,2,4]TRIAZINE-5(4H)-ACETAMIDES AS INHIBITORS OF THE NLRP3 INFLAMMASOME PATHWAY JANSSEN PHARMACEUTICA NV (BE) 2021-10-21 WO disclosed