SCHEMBL23950993

SCHEMBL23950993

O=CNc1ccc2nc(C(F)F)cn2c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.38
ALDH1A1 P00352 3/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 2/20 0.31
HPGD P15428 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
POLB P06746 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
CCNE2 O96020 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25241958 0.77 MCHR1 (0.47) MCHR1ALDH1A1SCN10AKDM4ENPC1
SCHEMBL2127565 0.75 ALDH1A3 (0.57) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL23950992 0.71 PIK3CG (0.38) MCHR1ALDH1A1SCN10AKDM4ENPC1
SCHEMBL23950206 0.70 MCHR1 (0.47) MCHR1ALDH1A1SCN10AKDM4ENPC1
SCHEMBL4441720 0.67 MEN1 (0.47) MCHR1ALDH1A1HPGDNFKB1
SCHEMBL12832006 0.62 SMN1; SMN2 (0.53) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL14701600 0.61 MCHR1 (0.59) MCHR1ALDH1A1SCN10AKDM4ENPC1
SCHEMBL469386 0.61 ALDH1A1 (0.72) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL90440 0.61 ALDH1A1 (0.56) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL21033162 0.61 KDM4E (0.40) MCHR1ALDH1A1KDM4ENPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021209552-A1 PYRAZOLO[1,5-D][1,2,4]TRIAZINE-5(4H)-ACETAMIDES AS INHIBITORS OF THE NLRP3 INFLAMMASOME PATHWAY JANSSEN PHARMACEUTICA NV (BE) 2021-10-21 WO disclosed