SCHEMBL23958683

SCHEMBL23958683

Cc1c(C(C)(C)NS(C)(=O)=O)cc(Cl)nc1-c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
PTGS2 P35354 13/20 0.37
SCN9A Q15858 1/20 0.37
PTGS1 P23219 3/20 0.36
DHODH Q02127 2/20 0.35
KDM4E B2RXH2 1/20 0.34
MITF O75030 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
STAT3 P40763 1/20 0.34
STAT1 P42224 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TLR9 Q9NR96 1/20 0.34
MAP2K4 P45985 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25686642 0.89 SCN9A (0.40) ADORA2AADORA1ADORA3ADORA2BPTGS2
SCHEMBL30007267 0.89 PTGS2 (0.38) ADORA2AADORA1ADORA3ADORA2BPTGS2
SCHEMBL23958629 0.89 PTGS2 (0.38) ADORA2AADORA1ADORA3ADORA2BPTGS2
SCHEMBL23958817 0.78 ADORA2A (0.42) ADORA2AADORA1ADORA3ADORA2BDHODH
SCHEMBL25686624 0.78 ADORA2A (0.39) ADORA2AADORA1ADORA3ADORA2BPTGS2
SCHEMBL23958624 0.75 PTGS2 (0.36) PTGS2SCN9AMAP2K4
SCHEMBL25686621 0.73 PTGDR2 (0.38) PTGS2LMNAMAP2K4
SCHEMBL23958600 0.72 CFTR (0.36) PTGS2SCN9APTGS1KDM4EMITF
SCHEMBL28909129 0.70 TRPV1 (0.34) PTGS2SCN9APTGS1
SCHEMBL23958852 0.70 CFTR (0.35) ADORA2AADORA1PTGS2SCN9APTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed