SCHEMBL23958828

SCHEMBL23958828

COC(=O)c1cc(Cl)nc(-c2ccc(F)cc2)c1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
CASP3 P42574 1/20 0.52
SENP8 Q96LD8 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
SENP6 Q9GZR1 1/20 0.52
DHODH Q02127 4/20 0.49
KDM4E B2RXH2 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
ALDH1A1 P00352 3/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
MAPT P10636 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
PLA2G2A P14555 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958825 0.89 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL30006707 0.88 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL23930037 0.88 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL25686480 0.85 LMNA (0.49) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL2513073 0.82 NPC1 (0.56) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL26791839 0.77 ALDH1A1 (0.41) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL23958849 0.76 NPC1 (0.56) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL18076802 0.75 KDM4E (0.44) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL30969925 0.75 KDM4E (0.44) SMN1; SMN2NPC1RAB9ACASP3SENP8
SCHEMBL2579354 0.75 LMNA (0.49) SMN1; SMN2NPC1RAB9ACASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed