SCHEMBL23966818

SCHEMBL23966818

COC(=O)Cn1nc(Cc2nc3cc(OCC(F)F)c(Cl)cc3[nH]2)c2c(F)ccc(F)c2c1=O

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 10/20 0.65
RHEB Q15382 3/20 0.38
F9 P00740 3/20 0.33
F10 P00742 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2C9 P11712 1/20 0.33
KCNH2 Q12809 1/20 0.33
TP53 P04637 1/20 0.33
EGFR P00533 1/20 0.33
BRS3 P32247 1/20 0.32
ENPP1 P22413 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23966815 0.92 S1PR2 (0.63) S1PR2RHEBCYP3A4CYP2C9
SCHEMBL23908839 0.92 S1PR2 (0.75) S1PR2RHEB
SCHEMBL23914704 0.92 S1PR2 (0.62) S1PR2RHEB
SCHEMBL23908779 0.86 S1PR2 (0.65) S1PR2RHEBTP53
SCHEMBL23966848 0.85 S1PR2 (0.72) S1PR2RHEBTP53EGFR
SCHEMBL23966844 0.78 S1PR2 (0.70) S1PR2RHEBCYP3A4CYP2C9
SCHEMBL23966531 0.77 S1PR2 (0.87) S1PR2CYP3A4CYP2C9TP53
SCHEMBL23908918 0.77 S1PR2 (0.69) S1PR2RHEB
SCHEMBL23915575 0.77 S1PR2 (0.69) S1PR2F9CYP3A4CYP2C9TP53
SCHEMBL23966552 0.77 S1PR2 (0.84) S1PR2RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed