SCHEMBL23967690

SCHEMBL23967690

CSc1ccc(-c2ccc(-c3nc4cc(CCCCC(=O)O)[nH]c4cc3Cl)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 10/20 0.46
PRKAB1 Q9Y478 10/20 0.46
PRKAA2 P54646 8/20 0.46
PRKAA1 Q13131 3/20 0.46
PRCP P42785 4/20 0.39
KDM4E B2RXH2 1/20 0.38
DHODH Q02127 1/20 0.36
S1PR1 P21453 1/20 0.36
PDE2A O00408 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
P2RY12 Q9H244 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23967843 0.97 PRKAG1 (0.47) PRKAG1PRKAB1PRKAA2PRKAA1PRCP
SCHEMBL16069385 0.85 PRKAG1 (0.45) PRKAG1PRKAB1PRKAA2PRKAA1PRCP
SCHEMBL16069390 0.82 PRKAG1 (0.46) PRKAG1PRKAB1PRKAA2PRKAA1PRCP
SCHEMBL23967847 0.82 PRKAG1 (0.47) PRKAG1PRKAB1PRKAA2PRKAA1S1PR1
SCHEMBL23967839 0.78 PRKAG1 (0.48) PRKAG1PRKAB1PRKAA2PRKAA1S1PR1
SCHEMBL16069387 0.73 SCD (0.41) PRKAG1PRKAB1PRKAA2
SCHEMBL16069386 0.72 SCD (0.41) PRKAG1PRKAB1PRKAA2
SCHEMBL17402606 0.72 PTGS2 (0.41)
SCHEMBL17402629 0.71 PTGS1 (0.42)
SCHEMBL16069513 0.70 SCD (0.39) PRKAG1PRKAB1PRKAA2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970119-B1 NOVEL INDOLE DERIVATIVES USEFUL AS ANTI-DIABETIC AGENTS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed