SCHEMBL23969765

SCHEMBL23969765

O=CNc1ccc(-c2cc(-c3ccccc3)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
KIF11 P52732 5/20 0.47
RXRA P19793 5/20 0.45
RXRG P48443 5/20 0.45
RXRB P28702 4/20 0.45
GLO1 Q04760 1/20 0.40
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40
KDR P35968 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
DHODH Q02127 1/20 0.39
P2RX1 P51575 1/20 0.39
PTPN1 P18031 1/20 0.39
BACE1 P56817 1/20 0.38
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23969869 0.87 ALDH1A1 (0.64) ALDH1A1PTPN1
SCHEMBL5429627 0.81 KIF11 (0.57) ALDH1A1KIF11
SCHEMBL14418354 0.81 ALDH1A1 (0.73) ALDH1A1DHODHPTPN1
SCHEMBL223423 0.81 ALDH1A1 (0.73) ALDH1A1DHODHPTPN1
SCHEMBL31093906 0.79 KIF11 (0.65) ALDH1A1KIF11RXRARXRGRXRB
SCHEMBL14471626 0.77 ALDH1A1 (0.60) ALDH1A1DHODHPTPN1
SCHEMBL28222642 0.77 KIF11 (0.70) ALDH1A1KIF11RXRARXRGRXRB
Nitrogen SCHEMBL27657438 0.75 KIF11 (0.60) ALDH1A1KIF11RXRARXRGRXRB
SCHEMBL183175 0.75 EPHX2 (0.52) ALDH1A1KIF11
SCHEMBL2138447 0.75 KIF11 (0.65) ALDH1A1KIF11RXRARXRGRXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353156-B1 TEAD TRANSCRIPTION FACTOR AUTOPALMITOYLATION INHIBITORS MASSACHUSETTS GEN HOSPITAL (US) 2021-11-03 EP disclosed