SCHEMBL23977436

SCHEMBL23977436

COc1ccc(C#N)cc1C#CS(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ESRRA P11474 1/20 0.39
KDM1A O60341 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
SLC6A4 P31645 1/20 0.37
ALPL P05186 1/20 0.37
IMPDH2 P12268 1/20 0.37
IMPDH1 P20839 1/20 0.37
ACLY P53396 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25909467 0.81 PTGDR2 (0.41) ARALDH1A1KDM4EPTGDR2
SCHEMBL2094284 0.81 ALDH1A1 (0.63) ARALDH1A1KDM4EUSP2ESRRA
SCHEMBL16951586 0.80 AR (0.49) ARALDH1A1KDM4EUSP2ESRRA
SCHEMBL1798639 0.77 AR (0.44) ARALDH1A1KDM4EUSP2ESRRA
SCHEMBL1798728 0.76 AR (0.49) ARALDH1A1KDM4EUSP2ESRRA
SCHEMBL1799535 0.75 AR (0.42) ARALDH1A1KDM4EUSP2KDM1A
SCHEMBL509522 0.73 AR (0.66) ARALDH1A1KDM4EUSP2KDM1A
SCHEMBL29490258 0.73 AR (0.66) ARALDH1A1KDM4EUSP2KDM1A
SCHEMBL4669307 0.72 ALDH1A1 (0.53) ARALDH1A1KDM4EUSP2ESRRA
SCHEMBL11616908 0.71 KDM1A (0.56) ARALDH1A1KDM4EUSP2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219813-A1 ANTIBACTERIAL AND ANTIFUNGAL PLEUROMUTILIN CONJUGATES SYDDANSK UNIVERSITET (DK) 2021-11-04 WO disclosed