SCHEMBL23978646

SCHEMBL23978646

COC(=O)[C@H](CNC(N)=O)NC(=O)c1c(Cl)ccc(Nc2ncc3ccccc3n2)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
INSR P06213 3/20 0.36
IGF1R P08069 3/20 0.36
ALK Q9UM73 3/20 0.36
FGFR1 P11362 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36
FGFR3 P22607 1/20 0.36
MAP3K5 Q99683 1/20 0.35
BRAF P15056 2/20 0.35
TAS1R3 Q7RTX0 5/20 0.34
TAS1R1 Q7RTX1 5/20 0.34
LRRK2 Q5S007 3/20 0.34
ITGB1 P05556 1/20 0.34
ITGA5 P08648 1/20 0.34
PIK3CG P48736 1/20 0.33
GSK3B P49841 1/20 0.33
CAMKK2 Q96RR4 1/20 0.33
TACR3 P29371 2/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979058 0.90 ITGB1 (0.39) MAP3K5ITGB1ITGA5
SCHEMBL23978630 0.84 FGFR1 (0.34) INSRIGF1RALKFGFR1FGFR2
SCHEMBL24804639 0.83 USP2 (0.41) TAS1R3TAS1R1
SCHEMBL30279406 0.83 USP2 (0.41) TAS1R3TAS1R1
SCHEMBL24804864 0.83 USP2 (0.41) TAS1R3TAS1R1
SCHEMBL23978706 0.78 MAP3K5 (0.45) IGF1RALKFGFR1FGFR2FGFR4
SCHEMBL23979049 0.76 P2RX3 (0.36) TAS1R3TAS1R1ITGB1ITGA5
SCHEMBL23978691 0.75 PRMT5 (0.36) TAS1R3TAS1R1ITGB1ITGA5
SCHEMBL23978642 0.75 LNPEP (0.39) TAS1R3TAS1R1ITGB1ITGA5
SCHEMBL23978627 0.75 MAP3K5 (0.44) IGF1RFGFR1FGFR2FGFR4FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed