SCHEMBL23979049

SCHEMBL23979049

COC(=O)[C@H](CNC(N)=O)NC(=O)c1c(Cl)ccc(Nc2cccc(C(C)C)c2)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.36
CA2 P00918 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
ITGB1 P05556 2/20 0.35
ITGA5 P08648 1/20 0.35
SYK P43405 1/20 0.35
PTGER3 P43115 1/20 0.34
FADS1 O60427 1/20 0.34
RAB9A P51151 1/20 0.34
ITGB2 P05107 2/20 0.33
ICAM1 P05362 2/20 0.33
ITGAL P20701 2/20 0.33
TAS1R3 Q7RTX0 4/20 0.33
TAS1R1 Q7RTX1 4/20 0.33
ITGA4 P13612 1/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978982 0.91 ITGAL (0.39) ITGB1ITGA5SYKPTGER3ITGB2
SCHEMBL23979060 0.81 USP2 (0.43) TAS1R3TAS1R1
SCHEMBL26493531 0.81 USP2 (0.43) TAS1R3TAS1R1
SCHEMBL24803327 0.81 USP2 (0.43) TAS1R3TAS1R1
SCHEMBL23979022 0.77 MAPT (0.41) P2RX3CA2PTGER3FADS1RAB9A
SCHEMBL23978642 0.76 LNPEP (0.39) ITGB1ITGA5ITGB2ICAM1ITGAL
SCHEMBL23978639 0.76 KCNQ2 (0.42) ITGB1ITGA5
SCHEMBL23978646 0.76 INSR (0.36) ITGB1ITGA5TAS1R3TAS1R1
SCHEMBL23979021 0.75 MEN1 (0.41) P2RX3CA2PTGER3FADS1SMN1; SMN2
SCHEMBL30337539 0.75 MEN1 (0.41) P2RX3CA2PTGER3FADS1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed