SCHEMBL23978654

SCHEMBL23978654

NC(=O)NC[C@H](NC(=O)c1c(Cl)ccc(NC(=O)CCc2ccccc2)c1Cl)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
ITGB1 P05556 4/20 0.42
ITGA5 P08648 4/20 0.42
ITGAV P06756 2/20 0.42
ITGA4 P13612 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 3/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 2/20 0.40
GAA P10253 1/20 0.40
ROCK2 O75116 1/20 0.40
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
HTT P42858 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978644 0.91 HPGD (0.45) ALDH1A1MEN1KMT2AALOX15MAPK1
SCHEMBL30279395 0.81 EPHX2 (0.49) ALDH1A1ITGB1ITGAVITGA4HTT
SCHEMBL26109531 0.81 EPHX2 (0.49) ALDH1A1ITGB1ITGAVITGA4HTT
SCHEMBL23978998 0.81 EPHX2 (0.49) ALDH1A1ITGB1ITGAVITGA4HTT
SCHEMBL23978657 0.81 EPHX2 (0.49) ALDH1A1ITGB1ITGAVITGA4HTT
SCHEMBL23978563 0.81 EPHX2 (0.49) ALDH1A1ITGB1ITGAVITGA4HTT
SCHEMBL24106071 0.79 ITGB1 (0.59) ITGB1ITGA5ITGAVITGA4ITGB2
SCHEMBL23979052 0.77 ITGB2 (0.39) ITGB1ITGA5ITGAVITGA4MEN1
SCHEMBL21376654 0.76 ITGB2 (0.59) ITGB1ITGA5ITGAVITGA4ITGB2
SCHEMBL23979071 0.75 ALDH1A1 (0.39) ALDH1A1ITGB1ITGA5ITGAVITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed