SCHEMBL23978682

SCHEMBL23978682

NC(=O)NC[C@H](NC(=O)c1c(Cl)ccc(N)c1Cl)C(=O)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 1/20 0.42
CASP3 P42574 1/20 0.41
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41
POLB P06746 2/20 0.40
MAPT P10636 6/20 0.39
S1PR4 O95977 3/20 0.39
S1PR1 P21453 2/20 0.39
ACE P12821 1/20 0.39
GAA P10253 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
TACR1 P25103 1/20 0.38
ALDH1A1 P00352 2/20 0.37
NTSR1 P30989 1/20 0.37
ATM Q13315 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978642 0.85 LNPEP (0.39) LNPEPITGB1ITGA5POLB
SCHEMBL24803388 0.81 EPHX2 (0.46) ALDH1A1
SCHEMBL30083836 0.81 EPHX2 (0.46) ALDH1A1
SCHEMBL26496578 0.81 EPHX2 (0.46) ALDH1A1
SCHEMBL23978981 0.79 POLB (0.48) CASP3POLBMAPTTACR1NPSR1
SCHEMBL30083853 0.79 SLC6A9 (0.35) LNPEPCASP3MAPTALDH1A1NTSR1
SCHEMBL24803374 0.79 SLC6A9 (0.35) LNPEPCASP3MAPTALDH1A1NTSR1
SCHEMBL23978717 0.79 SLC6A9 (0.35) LNPEPCASP3MAPTALDH1A1NTSR1
SCHEMBL23978763 0.78 ITGB1 (0.46) CASP3ITGB1ITGA5POLBMAPT
SCHEMBL23978762 0.77 ITGB2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed