SCHEMBL23978987

SCHEMBL23978987

CC(C)(C)OC(=O)NC[C@H](CCC(=O)c1c(Cl)ccc(NC(=O)Cc2cccc(Cl)c2)c1Cl)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.40
KCNQ2 O43526 4/20 0.39
GLS O94925 4/20 0.36
KDM4E B2RXH2 1/20 0.36
SYK P43405 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 2/20 0.35
ANO1 Q5XXA6 1/20 0.35
MAPK8 P45983 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1C Q13936 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978812 0.84 CTSL (0.45) CTSLKCNQ2GLSKDM4ESYK
SCHEMBL26103779 0.84 CTSL (0.45) CTSLKCNQ2GLSKDM4ESYK
SCHEMBL30279367 0.84 CTSL (0.45) CTSLKCNQ2GLSKDM4ESYK
SCHEMBL23979131 0.80 KCNQ2 (0.39) KCNQ2MEN1KMT2AALDH1A1MAPK8
SCHEMBL24805443 0.78 CTSL (0.43) CTSLKCNQ2GLSKDM4EANO1
SCHEMBL23978985 0.76 SLC1A3 (0.38) KCNQ2GLSMEN1KMT2A
SCHEMBL1185574 0.74 CTSL (0.59) CTSLKDM4ESYKMEN1KMT2A
SCHEMBL30336898 0.73 KCNQ2 (0.54) KCNQ2KDM4EMEN1KMT2AALDH1A1
SCHEMBL23978834 0.73 KCNQ2 (0.54) KCNQ2KDM4EMEN1KMT2AALDH1A1
SCHEMBL23978894 0.72 KCNQ2 (0.54) KCNQ2MEN1KMT2AALDH1A1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed