SCHEMBL23978985

SCHEMBL23978985

NC(=O)NC[C@H](CCC(=O)c1c(Cl)ccc(NC(=O)Cc2ccc(F)c(Cl)c2)c1Cl)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
PIK3CA P42336 1/20 0.36
KCNJ6 P48051 1/20 0.34
KCNJ5 P48544 1/20 0.34
KCNJ3 P48549 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
KCNQ2 O43526 1/20 0.32
GLS O94925 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979131 0.78 KCNQ2 (0.39) MEN1KMT2ALMNAMAPTKCNQ2
SCHEMBL23978694 0.78 CA12 (0.46) SLC1A3SLC1A2SLC1A1CA12CA1
SCHEMBL23978987 0.76 CTSL (0.40) MEN1KMT2AKCNQ2GLS
SCHEMBL26497251 0.65 KCNQ2 (0.38) CA1CA2KCNJ5KCNJ3MEN1
SCHEMBL23978667 0.65 SMN1; SMN2 (0.48) MEN1KMT2ALMNAMAPTHTT
SCHEMBL23978639 0.65 KCNQ2 (0.42) MEN1KMT2AKCNQ2
SCHEMBL23978676 0.64 KDM4E (0.33) KMT2ALMNA
SCHEMBL23978834 0.64 KCNQ2 (0.54) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL30336898 0.64 KCNQ2 (0.54) CA1CA2MEN1KMT2AL3MBTL1
SCHEMBL23978654 0.63 ALDH1A1 (0.42) MEN1KMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed