SCHEMBL23980604

SCHEMBL23980604

COc1ccc2ccc(SC)cc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.59
CYP2A6 P11509 1/20 0.59
CYP1A1 P04798 6/20 0.55
CYP1B1 Q16678 6/20 0.55
RAB9A P51151 1/20 0.50
HSD17B1 P14061 1/20 0.47
HSD17B2 P37059 1/20 0.47
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
KMT2A Q03164 1/20 0.46
SLC6A4 P31645 1/20 0.45
KDM4E B2RXH2 1/20 0.44
GSTP1 P09211 1/20 0.44
HTR1A P08908 1/20 0.44
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
CYP17A1 P05093 1/20 0.44
CYP11B2 P19099 1/20 0.44
NCF1 P14598 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502871 0.96 CYP1A2 (0.59) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL443528 0.84 CYP2A6 (0.80) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL29367032 0.84 CYP2A6 (0.80) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL29740639 0.82 AKR1C3 (0.45) CYP1A2CYP2A6SLC6A4KDM4E
SCHEMBL21551821 0.82 AKR1C3 (0.45) CYP1A2CYP2A6SLC6A4KDM4E
SCHEMBL23980770 0.81 CYP1A1 (0.47) CYP1A2CYP1A1CYP1B1RAB9A
SCHEMBL7763044 0.80 CYP2A6 (0.60) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL7760649 0.80 CYP1A2 (0.60) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL6891918 0.79 CYP1A2 (0.71) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A
SCHEMBL7456084 0.79 CYP1A2 (0.71) CYP1A2CYP2A6CYP1A1CYP1B1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230234925-A1 GPR52 MODULATORS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. 2023-07-27 US disclosed
WO-2021222542-A1 5-AMINO-2-PIPERIDINON-3-YL-1-OXOISOINDOLINE DERIVATIVES FOR DEGRADATION OF IKZF2 DEGRADERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2021-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230234925-A1 GPR52 MODULATORS AND METHODS OF USE GPR52, GPR68, GPR35 CYP1A2 1058/4885CYP2A6 1030/4885CYP1A1 2102/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.