SCHEMBL24006703

SCHEMBL24006703

C=C(C)c1ccc(F)cc1C(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.38
RECQL P46063 1/20 0.36
CES2 O00748 4/20 0.35
CES1 P23141 4/20 0.35
MAPK14 Q16539 2/20 0.32
PSEN1 P49768 2/20 0.32
PSEN2 P49810 2/20 0.32
APH1B Q8WW43 2/20 0.32
NCSTN Q92542 2/20 0.32
APH1A Q96BI3 2/20 0.32
PSENEN Q9NZ42 2/20 0.32
P2RX7 Q99572 1/20 0.32
GCGR P47871 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RXRA P19793 1/20 0.31
TRPA1 O75762 1/20 0.31
LMNA P02545 1/20 0.31
CHRM1 P11229 1/20 0.31
SLC6A2 P23975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24006702 0.83 RECQL (0.35) HRH4RECQLCES2CES1MAPK14
SCHEMBL24007928 0.79 HRH4 (0.38) HRH4RECQLMAPK14
SCHEMBL1408588 0.78 ACE2 (0.38) RXRATRPA1LMNACHRM1SLC6A2
SCHEMBL7912361 0.78 CA1 (0.37) CES2MEN1KMT2ATRPA1LMNA
SCHEMBL21207989 0.77 CES2 (0.41) HRH4CES2CES1
SCHEMBL7288273 0.77 KEAP1 (0.48) RECQLCES2CES1
SCHEMBL7281400 0.76 CES2 (0.42) RECQLCES2CES1MAPK14PSEN1
SCHEMBL13689710 0.75 CES2 (0.56) CES2CES1MEN1KMT2A
SCHEMBL29727310 0.75 CES2 (0.56) CES2CES1MEN1KMT2A
SCHEMBL13651368 0.75 GCGR (0.37) HRH4RECQLGCGRRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021226208-A2 HETEROAROMATIC MACROCYCLIC ETHER CHEMOTHERAPEUTIC AGENTS NUVALENT, INC. (US) 2021-11-11 WO disclosed