SCHEMBL24006702

SCHEMBL24006702

C=C(N)c1ccc(F)cc1C(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.35
HRH4 Q9H3N8 2/20 0.35
CES2 O00748 3/20 0.34
CES1 P23141 3/20 0.34
MAPK14 Q16539 1/20 0.34
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
KEAP1 Q14145 1/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
P2RX7 Q99572 1/20 0.31
GCGR P47871 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24006703 0.83 HRH4 (0.38) RECQLHRH4CES2CES1MAPK14
SCHEMBL24007928 0.80 HRH4 (0.38) RECQLHRH4MAPK14
SCHEMBL24006762 0.80 HRH4 (0.37) RECQLHRH4CES2CES1MAPK14
SCHEMBL7288273 0.76 KEAP1 (0.48) RECQLCES2CES1KEAP1
SCHEMBL7281400 0.74 CES2 (0.42) RECQLCES2CES1MAPK14KEAP1
SCHEMBL19519579 0.74 GABRA1 (0.48) NOS3NOS1
SCHEMBL24006646 0.74 HRH4 (0.33) RECQLHRH4MAPK14
SCHEMBL24007412 0.73 HRH4 (0.39) HRH4CES2CES1KEAP1NOS3
SCHEMBL18375724 0.71 SLC6A4 (0.45) RECQLCES2CES1
SCHEMBL12197672 0.71 CYP1A2 (0.39) RECQLHRH4CES2CES1PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021226208-A2 HETEROAROMATIC MACROCYCLIC ETHER CHEMOTHERAPEUTIC AGENTS NUVALENT, INC. (US) 2021-11-11 WO disclosed