SCHEMBL24019772

SCHEMBL24019772

CC(C)NC(=O)c1cc2cc(F)cc(Cl)c2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.53
ALPL P05186 2/20 0.45
SETD2 Q9BYW2 1/20 0.41
AR P10275 1/20 0.39
HRH4 Q9H3N8 3/20 0.39
EIF4A3 P38919 1/20 0.37
CTNNB1 P35222 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RECQL P46063 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
PYGL P06737 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24019966 0.87 ALOX15 (0.58) ALOX15ALPLHRH4CTNNB1SMN1; SMN2
SCHEMBL24019691 0.83 ALOX15 (0.51) ALOX15ALPLHRH4CTNNB1NPC1
SCHEMBL25758841 0.83 XDH (0.49) ALOX15ALPLSETD2ARHRH4
SCHEMBL24019964 0.81 ALOX15 (0.58) ALOX15ALPLAREIF4A3POLB
SCHEMBL25768433 0.80 ALOX15 (0.53) ALOX15HRH4MEN1KMT2A
SCHEMBL24019959 0.80 ALOX15 (0.57) ALOX15ALPLSETD2HRH4PYGL
SCHEMBL24019763 0.79 ALOX15 (0.52) ALOX15ALPLAREIF4A3MEN1
SCHEMBL25812181 0.79 HRH4 (0.43) HRH4EIF4A3MEN1NPC1POLB
SCHEMBL24740347 0.78 ALOX15 (0.61) ALOX15ALPLARHRH4EIF4A3
SCHEMBL24019762 0.77 ALOX15 (0.60) ALOX15ALPLEIF4A3POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-07-06 US disclosed
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. 2023-07-06 US disclosed
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2022-12-13 US disclosed
US-11174231-B1 Inhibitors of cysteine proteases and methods of use thereof Pardes Biosciences, Inc. (US) 2021-11-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11174231-B1 Inhibitors of cysteine proteases and methods of use thereof CTRL, CTSV, CTSL ALOX15 1749/4885ALPL 1768/4885SETD2 2742/4885
US-11524940-B1 Inhibitors of cysteine proteases and methods of use thereof CTRL, CTSV, CTSL ALOX15 1749/4885ALPL 1768/4885SETD2 2742/4885
US-20230212152-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF CTRL, CTSL, CTSV ALOX15 1455/4885ALPL 1886/4885SETD2 2786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.