SCHEMBL24034825

SCHEMBL24034825

Cc1nnn(-c2ccc(Cl)cc2)c1CN1CC=C(N(C)C)C=N1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.38
NOTUM Q6P988 1/20 0.36
PTGS2 P35354 4/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HTT P42858 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
RAB9A P51151 1/20 0.33
P2RX7 Q99572 1/20 0.32
TP53 P04637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
KCNH2 Q12809 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24098476 0.68 NOTUM (0.50) MAPTNOTUMPTGS2CYP1A2CYP2C19
SCHEMBL21834180 0.68 NOTUM (0.62) MAPTNOTUMPTGS2CYP1A2CYP2C19
SCHEMBL10091953 0.63 NOTUM (0.62) MAPTNOTUMPTGS2CYP1A2CYP2C19
SCHEMBL25045396 0.62 GABRA5 (0.44) NOTUMPTGS2CYP1A2CYP2C19CYP2D6
SCHEMBL25045387 0.60 KMT2A (0.56) MAPTNOTUMPTGS2CYP2C9CA1
SCHEMBL30237036 0.59 GABRA5 (0.39) NOTUMPTGS2CYP1A2CYP2C19CYP2D6
SCHEMBL28906183 0.59 ALDH1A1 (0.54) MAPTNOTUMPTGS2CA1CA2
SCHEMBL9730309 0.57 PTGS2 (0.45) PTGS2CYP1A2RAB9ATP53ALDH1A1
SCHEMBL25044741 0.56 ALDH1A1 (0.49) MAPTNOTUMCYP1A2CYP2C19CYP2C9
SCHEMBL25044752 0.55 GABRA5 (0.44) ALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021228795-A1 NEW TRIAZOLYL DERIVATIVES AS GABA A ALPHA5 PAM F. HOFFMANN-LA ROCHE AG (CH) 2021-11-18 WO disclosed