SCHEMBL9730309

SCHEMBL9730309

Cc1nnn(-c2ccc(F)cc2)c1CCl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.45
GABRA5 P31644 8/20 0.43
GABRG2 P18507 5/20 0.43
GABRB3 P28472 5/20 0.43
KCNH2 Q12809 2/20 0.43
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DCTPP1 Q9H773 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
TP53 P04637 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2683661 0.83 PTGS2 (0.49) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL21834124 0.83 GABRA5 (0.46) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL9730918 0.80 PTGS2 (0.39) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL12530467 0.77 PTGS2 (0.60) PTGS2ALDH1A1LMNADCTPP1MEN1
SCHEMBL2688352 0.74 GABRA5 (0.54) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL30282901 0.74 GABRA5 (0.54) PTGS2GABRA5GABRG2GABRB3KCNH2
Hydrochloric Acid SCHEMBL9731318 0.74 DCTPP1 (0.41) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL30237887 0.71 GABRA5 (0.52) PTGS2GABRA5GABRG2GABRB3KCNH2
SCHEMBL23116877 0.71 MAPT (0.49) ALDH1A1NPSR1L3MBTL1MEN1KMT2A
SCHEMBL21834180 0.70 NOTUM (0.62) PTGS2ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081136-A 1,2,3-TRIAZOLE COMPOUNDS ACTIVE AS INHIBITORS OF THE ENZYME HMG-COA REDUCTASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ZAMBON GROUP S.P.A. (IT) 1992-01-14 US disclosed
EP-0433842-A2 1,2,3-Triazole derivatives active as inhibitors of the enzyme HMG-COA reductase and pharmaceutical compositions containing them ZAMBON GROUP S.p.A. (IT) 1991-06-26 EP disclosed