SCHEMBL2407202

SCHEMBL2407202

O=C(O)N(CCC1CCN(c2cccc(-c3ccc(F)cc3)n2)CC1)Cc1cncs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
CYP2C9 P11712 2/20 0.38
HSD11B1 P28845 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
DRD3 P35462 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CNR1 P21554 1/20 0.36
FFAR4 Q5NUL3 4/20 0.36
MCHR1 Q99705 2/20 0.35
ENPP2 Q13822 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2406938 0.85 DGAT1 (0.39) CKS1BSKP1SKP2HTR1ADRD4
SCHEMBL2407375 0.84 CKS1B (0.40) CKS1BSKP1SKP2HTR1ADRD2
SCHEMBL2405880 0.83 CKS1B (0.40) CKS1BSKP1SKP2HTR1ADRD2
SCHEMBL2406177 0.83 PDE10A (0.40) CKS1BSKP1SKP2CYP3A4
SCHEMBL2405423 0.83 PDE10A (0.42) CKS1BSKP1SKP2HTR1A
SCHEMBL1728786 0.82 HTR1A (0.42) CKS1BSKP1SKP2CYP2C9HTR1A
SCHEMBL2407608 0.76 HRH3 (0.43) HTR1AMCHR1
SCHEMBL2407363 0.76 CNR1 (0.37) CYP2C9HSD11B1NPC1RAB9ACNR1
SCHEMBL1710840 0.76 HTR1A (0.47) CKS1BSKP1SKP2CYP2C9HSD11B1
SCHEMBL2411396 0.75 CHRM4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8912218-B2 Alkylthiazol carbamate derivatives, preparation thereof and therapeutic use thereof SANOFI (FR) 2014-12-16 US disclosed
US-20110212963-A1 ALKYLTHIAZOL CARBAMATE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212963-A1 ALKYLTHIAZOL CARBAMATE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF MET, ALK, REL CKS1B 2188/4885SKP1 3476/4885SKP2 3826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.