SCHEMBL2407589

SCHEMBL2407589

CC(C)(C)CN(Cc1cn(S(=O)(=O)c2cccc(S(C)(=O)=O)c2)c(-c2cccnc2F)c1F)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.39
PTGDR2 Q9Y5Y4 10/20 0.37
CCKAR P32238 1/20 0.32
PIP4K2A P48426 1/20 0.31
PIP4K2C Q8TBX8 1/20 0.31
PTGS2 P35354 1/20 0.31
PDE4A P27815 3/20 0.31
PDE4B Q07343 3/20 0.31
PDE4C Q08493 3/20 0.31
PDE4D Q08499 3/20 0.31
OXTR P30559 1/20 0.30
CHRM5 P08912 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4420273 0.92 HTR6 (0.36) PTGDR2CCKARHTR6
SCHEMBL2411936 0.90 EPHX2 (0.33) PTGDR2CCKAR
SCHEMBL2415890 0.90 GAA (0.32) PTGDR2CCKAR
SCHEMBL2409039 0.90 RXFP1 (0.33) PTGDR2CCKAR
SCHEMBL2411542 0.90 MET (0.41) METPTGDR2CHRM5HTR6
SCHEMBL2410118 0.89 PPME1 (0.35) PTGDR2HTR6
SCHEMBL2411045 0.88 PTGER2 (0.33) PTGDR2HTR6
SCHEMBL2408493 0.88 GAA (0.30) PTGDR2
SCHEMBL2409445 0.87 ESR1 (0.39) PTGDR2CCKARHTR6
SCHEMBL5003157 0.87 MET (0.41) METPTGDR2CCKARPIP4K2APIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed