SCHEMBL2409445

SCHEMBL2409445

CC(C)(C)CN(Cc1cn(S(=O)(=O)c2ccc(O)cc2)c(-c2cccnc2F)c1F)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
PTGDR2 Q9Y5Y4 10/20 0.33
HTR6 P50406 2/20 0.32
CCKAR P32238 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP8 P22894 1/20 0.31
MMP13 P45452 1/20 0.31
GPR55 Q9Y2T6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4424130 0.94 ESR1 (0.34) ESR1PTGDR2
SCHEMBL1833794 0.90 PTGDR2 (0.34) PTGDR2CCKARMMP2MMP9MMP8
SCHEMBL2411210 0.89 HTR6 (0.38) HTR6MMP9MMP8MMP13
SCHEMBL2411045 0.89 PTGER2 (0.33) PTGDR2HTR6
SCHEMBL4420273 0.88 HTR6 (0.36) PTGDR2HTR6CCKAR
SCHEMBL1834429 0.88 PTGDR2 (0.32) PTGDR2CCKAR
SCHEMBL4570003 0.88 TAS2R14 (0.35) PTGDR2MMP2MMP9MMP8MMP13
SCHEMBL2408899 0.87 PTGDR2 (0.30) PTGDR2
SCHEMBL2407589 0.87 MET (0.39) PTGDR2HTR6CCKAR
SCHEMBL2413762 0.87 SLC6A9 (0.35) PTGDR2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed