SCHEMBL2407592

SCHEMBL2407592

N#Cc1c(F)cccc1-c1ccc(C(=O)N2CCc3ncnc(N4CCC(C(=O)C5CC5)CC4)c3C2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.55
KCNK9 Q9NPC2 1/20 0.55
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
GRM5 P41594 2/20 0.35
GRM1 Q13255 4/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
IDH1 O75874 1/20 0.34
LRRK2 Q5S007 2/20 0.33
PARP1 P09874 1/20 0.33
KDM1A O60341 1/20 0.33
ABL1 P00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12320839 0.88 KCNK3 (0.57) KCNK3KCNK9CDK4CCND1GRM5
SCHEMBL2407799 0.83 KCNK3 (0.65) KCNK3KCNK9CDK4CCND1GRM5
SCHEMBL12320837 0.79 KCNK3 (0.61) KCNK3KCNK9GRM5HPGDHTT
SCHEMBL2407040 0.74 KCNK3 (0.87) KCNK3KCNK9MEN1ALDH1A1HPGD
SCHEMBL30664070 0.71 KCNK3 (1.00) KCNK3KCNK9MEN1ALDH1A1HPGD
SCHEMBL2406138 0.71 KCNK3 (1.00) KCNK3KCNK9MEN1ALDH1A1HPGD
SCHEMBL2410232 0.70 KCNK3 (0.72) KCNK3KCNK9CDK4CCND1MAPT
SCHEMBL2410478 0.70 KCNK3 (0.73) KCNK3KCNK9MEN1ALDH1A1KMT2A
SCHEMBL2407042 0.68 KCNK3 (0.68) KCNK3KCNK9MEN1ALDH1A1KMT2A
SCHEMBL2406140 0.67 KCNK3 (0.66) KCNK3KCNK9MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed