SCHEMBL2408335

SCHEMBL2408335

O=C(Cc1ccccc1)OC1CCN(CCc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.61
HTR2A P28223 2/20 0.57
OPRM1 P35372 2/20 0.56
OPRD1 P41143 2/20 0.56
OPRK1 P41145 2/20 0.56
ACHE P22303 1/20 0.54
CCR3 P51677 1/20 0.52
DRD2 P14416 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10969939 0.86 HTR2A (0.54) SIGMAR1HTR2AOPRM1OPRD1OPRK1
SCHEMBL7276778 0.85 SIGMAR1 (0.54) SIGMAR1HTR2AOPRM1OPRD1ACHE
SCHEMBL13266074 0.84 ALDH1A1 (0.64) HTR2AOPRM1OPRK1HTR2CHTR2B
SCHEMBL27474479 0.81 TP53 (0.50)
SCHEMBL15147383 0.79 CHRM3 (0.60)
SCHEMBL10874959 0.79 STS (0.48)
SCHEMBL15147380 0.79 CHRM3 (0.60)
SCHEMBL6761969 0.79 CYP19A1 (0.66)
SCHEMBL5049441 0.79 CYP19A1 (0.71)
SCHEMBL5709472 0.77 HTR2A (0.50) SIGMAR1HTR2AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150196522-A1 METHODS OF USING (1S,3S)-3-AMINO-4-DIFLUOROMETHYLENYL-1-CYCLOPENTANOIC ACID NORTHWESTERN UNIVERSITY 2015-07-16 US disclosed
US-8969413-B2 Methods of using (1S,3S)-3-amino-4-difluoromethylenyl-1-cyclopentanoic acid CATALYST PHARMACEUTICAL PARTNERS (US) 2015-03-03 US disclosed
US-20130041028-A1 METHODS OF USING (1S,3S)-3-AMINO-4-DIFLUOROMETHYLENYL-1-CYCLOPENTANOIC ACID NORTHWESTERN UNIVERSITY (US) 2013-02-14 US disclosed
EP-2542234-A2 METHODS OF USING (1S, 3S) -3-AMINO-4-DIFLUOROMETHYLENYL-1-CYCLOPENTANOIC ACID North Western University (US) 2013-01-09 EP disclosed
WO-2011106692-A2 METHODS OF USING (1S, 3S) -3-AMINO-4-DIFLUOROMETHYLENYL-1-CYCLOPENTANOIC ACID NORTHWESTERN UNIVERSITY (US) 2011-09-01 WO disclosed