SCHEMBL2408757

SCHEMBL2408757

CN(Cc1c[nH]c(-c2cccnc2C(F)(F)F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.41
CACNA1G O43497 1/20 0.38
CACNA1B Q00975 1/20 0.38
CACNA1C Q13936 1/20 0.38
SSTR4 P31391 2/20 0.37
PDK2 Q15119 1/20 0.36
TACR1 P25103 2/20 0.35
HTR2C P28335 6/20 0.34
SLC6A4 P31645 6/20 0.34
IDO1 P14902 1/20 0.34
HTR2A P28223 1/20 0.34
RIPK1 Q13546 2/20 0.33
PTK2 Q05397 1/20 0.32
NTRK1 P04629 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830977 0.89 SSTR4 (0.38) SOS1CACNA1GCACNA1BCACNA1CSSTR4
SCHEMBL2409140 0.87 POLB (0.36) SOS1CACNA1GCACNA1BCACNA1CSSTR4
SCHEMBL4416056 0.86 TACR1 (0.36) SSTR4TACR1RIPK1NTRK1
SCHEMBL2410739 0.84 PLCG1 (0.37) SOS1CACNA1GCACNA1BCACNA1CSSTR4
SCHEMBL2408759 0.80 DHODH (0.33) SSTR4TACR1SLC6A4NTRK1
SCHEMBL2407583 0.76 SOS1 (0.36) SOS1SSTR4PDK2TACR1HTR2C
SCHEMBL2408643 0.74 SOS1 (0.33) SOS1SSTR4PDK2TACR1HTR2C
SCHEMBL2194154 0.73 NAPRT (0.38) TACR1RIPK1
SCHEMBL2409767 0.73 HTR2C (0.38) CACNA1GCACNA1BCACNA1CSSTR4PDK2
SCHEMBL30439835 0.73 IDO1 (0.42) SOS1CACNA1GCACNA1BCACNA1CPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed