SCHEMBL2408759

SCHEMBL2408759

CC(C)(C)CN(Cc1c[nH]c(-c2cccnc2C(F)(F)F)c1F)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.33
NTRK1 P04629 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SSTR4 P31391 1/20 0.31
FFAR4 Q5NUL3 1/20 0.30
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830980 0.89 NAPRT (0.33) DHODHNTRK1FFAR4
SCHEMBL2416412 0.87 DHODH (0.32) DHODHNTRK1FFAR4
SCHEMBL4416056 0.86 TACR1 (0.36) DHODHNTRK1SSTR4FFAR4TACR1
SCHEMBL2410567 0.84 PLCG1 (0.35)
SCHEMBL2408757 0.80 SOS1 (0.41) NTRK1SLC6A4SSTR4TACR1
SCHEMBL2407587 0.75 DHODH (0.34) DHODH
SCHEMBL2408755 0.75 WDR5 (0.33) DHODHSSTR4
SCHEMBL4416060 0.74 MTNR1A (0.42) DHODH
SCHEMBL2194154 0.73 NAPRT (0.38) DHODHFFAR4TACR1
SCHEMBL2408646 0.73 RORC (0.33) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed