SCHEMBL2407583

SCHEMBL2407583

CN(Cc1cn(S(=O)(=O)c2ccccc2)c(-c2cccnc2C(F)(F)F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.36
HTR6 P50406 6/20 0.34
HTR2C P28335 4/20 0.33
SLC6A4 P31645 4/20 0.33
DHODH Q02127 1/20 0.33
PDK2 Q15119 1/20 0.33
F2 P00734 2/20 0.33
TNFSF11 O14788 1/20 0.33
SSTR4 P31391 1/20 0.32
TACR1 P25103 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2408643 0.93 SOS1 (0.33) SOS1HTR6HTR2CSLC6A4PDK2
SCHEMBL4999141 0.90 HTR6 (0.37) HTR6DHODHTNFSF11TACR1PTGDR2
SCHEMBL2412417 0.89 HTR2C (0.35) HTR6HTR2CSLC6A4F2TNFSF11
SCHEMBL2409996 0.87 HTR6 (0.33) HTR6HTR2CSLC6A4PDK2F2
SCHEMBL2409441 0.85 HTR2C (0.35) HTR6HTR2CSLC6A4PDK2F2
SCHEMBL2411042 0.84 HTR6 (0.33) HTR6HTR2CSLC6A4F2SSTR4
SCHEMBL4420269 0.83 HTR6 (0.37) HTR6HTR2CSLC6A4F2HTR2A
SCHEMBL2411207 0.83 HTR6 (0.39) HTR6HTR2CSLC6A4
SCHEMBL2407587 0.83 DHODH (0.34) HTR6DHODHPTGDR2
SCHEMBL5005875 0.83 HTR6 (0.35) HTR6DHODHTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed