SCHEMBL2408643

SCHEMBL2408643

CN(Cc1cn(S(=O)(=O)c2cccnc2)c(-c2cccnc2C(F)(F)F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.33
GPBAR1 Q8TDU6 4/20 0.33
PTK2 Q05397 1/20 0.32
RORC P51449 2/20 0.31
HTR6 P50406 1/20 0.31
SSTR4 P31391 1/20 0.31
TACR1 P25103 1/20 0.31
POLQ O75417 1/20 0.30
HTR2C P28335 2/20 0.30
SLC6A4 P31645 2/20 0.30
PDK2 Q15119 1/20 0.30
HTR2A P28223 1/20 0.30
F2 P00734 1/20 0.30
KAT8 Q9H7Z6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2407583 0.93 SOS1 (0.36) SOS1HTR6SSTR4TACR1HTR2C
SCHEMBL2411042 0.92 HTR6 (0.33) GPBAR1PTK2RORCHTR6SSTR4
SCHEMBL2410573 0.90 GPBAR1 (0.34) GPBAR1HTR6HTR2CSLC6A4HTR2A
SCHEMBL5005875 0.89 HTR6 (0.35) GPBAR1RORCHTR6TACR1POLQ
SCHEMBL2408006 0.88 PLCG1 (0.32) HTR6KAT8
SCHEMBL2408646 0.83 RORC (0.33) GPBAR1RORCHTR6
SCHEMBL1832149 0.83 HTR2C (0.33) GPBAR1RORCHTR2CSLC6A4PDK2
SCHEMBL1833792 0.83 KAT6A (0.32) SSTR4HTR2CSLC6A4HTR2AF2
SCHEMBL1832665 0.82 RORC (0.35) GPBAR1RORCHTR2CSLC6A4PDK2
SCHEMBL4999141 0.82 HTR6 (0.37) HTR6TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed