SCHEMBL24089946

SCHEMBL24089946

CN(C)Cc1cccc(Nc2nc3ccccc3c(=O)n2-c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 3/20 0.49
MAPT P10636 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
USP2 O75604 1/20 0.45
PDE7A Q13946 1/20 0.45
ALDH1A1 P00352 1/20 0.44
TOP2A P11388 1/20 0.44
TOP2B Q02880 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29623228 1.00 ACP1 (0.49) ACP1MAPTNPC1RAB9AUSP2
SCHEMBL24090098 0.89 TDO2 (0.49) ACP1ALDH1A1
SCHEMBL24090011 0.89 ACP1 (0.50) ACP1
SCHEMBL24090135 0.88 USP2 (0.48) ACP1MAPTNPC1RAB9AUSP2
SCHEMBL24090012 0.86 TOP2A (0.60) MAPTNPC1RAB9AUSP2PDE7A
SCHEMBL24089906 0.81 ACP1 (0.50) ACP1MAPTNPC1RAB9AUSP2
SCHEMBL24089947 0.79 ALOX12 (0.55) MAPTRAB9AUSP2PDE7A
SCHEMBL24089969 0.79 IDO1 (0.42) ACP1MAPTUSP2PDE7A
SCHEMBL23045341 0.78 ACP1 (0.48) ACP1NPC1
SCHEMBL24090006 0.78 TDO2 (0.51) ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352366-B2 2-aminoquinazolinone derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-06-07 US disclosed
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-05-12 US disclosed
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, CRKL ACP1 3959/4885MAPT 4827/4885NPC1 1269/4885
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, SLC26A3 ACP1 4435/4885MAPT 4783/4885NPC1 1276/4885
US-11352366-B2 2-aminoquinazolinone derivative CNKSR1, HAX1, SLC26A3 ACP1 4435/4885MAPT 4783/4885NPC1 1276/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.