SCHEMBL24093147

SCHEMBL24093147

CSNc1cccc(CN(C)C)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
NOS1 P29475 3/20 0.44
NOS2 P35228 1/20 0.44
HPGD P15428 1/20 0.41
KDM1A O60341 1/20 0.40
RCOR1 Q9UKL0 1/20 0.40
HTR7 P34969 2/20 0.40
ACP1 P24666 3/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
ACHE P22303 1/20 0.37
TAAR1 Q96RJ0 2/20 0.37
HRH3 Q9Y5N1 1/20 0.36
POLB P06746 1/20 0.36
HTR6 P50406 1/20 0.36
KIT P10721 1/20 0.34
PDGFRA P16234 1/20 0.34
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6175219 0.79 TSHR (0.50) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL30704883 0.78 NOS1 (0.49) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL4200353 0.78 NOS1 (0.49) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL7258875 0.76 ALDH1A1 (0.47) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL23134330 0.76 NOS1 (0.51) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL989636 0.76 ALDH1A1 (0.67) ALDH1A1TSHRNOS1HPGDHTR7
SCHEMBL15034736 0.75 ALDH1A1 (0.45) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL23133807 0.75 ALDH1A1 (0.45) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL23134425 0.71 ALDH1A1 (0.48) ALDH1A1TSHRNOS1NOS2HPGD
SCHEMBL3728364 0.71 NOS1 (0.50) ALDH1A1TSHRNOS1NOS2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3452464-B1 PYRAZOLE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USE THEREOF HOFFMANN LA ROCHE (CH) 2021-12-15 EP disclosed