SCHEMBL24095946

SCHEMBL24095946

CN(CCc1ccc(O)cc1)C(=O)CCC(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 1/20 0.49
CA2 P00918 1/20 0.44
OPRM1 P35372 2/20 0.44
OPRD1 P41143 2/20 0.44
OPRK1 P41145 2/20 0.44
LTB4R Q15722 5/20 0.44
LTB4R2 Q9NPC1 5/20 0.44
CDK8 P49336 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
KDM4E B2RXH2 3/20 0.39
F13A1 P00488 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
SLC6A2 P23975 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4319665 0.81 KMT2A (0.64) ESRRGOPRM1OPRD1OPRK1LTB4R
SCHEMBL3999705 0.76 CDK8 (0.74) CDK8CLK4KMT2ANPC1RAB9A
SCHEMBL8758089 0.76 ESRRG (0.56) ESRRGCA2OPRM1OPRD1OPRK1
SCHEMBL154384 0.75 CA2 (0.61) CA2KMT2AESR1ESR2KDM4E
SCHEMBL26294033 0.75 ESRRG (0.49) ESRRGCA2OPRM1OPRD1OPRK1
SCHEMBL4324200 0.74 KMT2A (0.46) ESRRGOPRM1OPRD1OPRK1CDK8
SCHEMBL23732700 0.74 TMEM97 (0.54) ESRRGOPRM1OPRD1OPRK1CDK8
SCHEMBL934532 0.74 CA2 (0.59) CA2KMT2AESR1ESR2KDM4E
Butane SCHEMBL10453910 0.73 CA2 (0.53) CA2KMT2AESR1ESR2KDM4E
SCHEMBL4938894 0.72 ACHE (0.57) CA2LTB4RKMT2AESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252640-A1 ASPARAGINE DERIVATIVES AND METHODS OF USING SAME SENDA BIOSCIENCES, INC. (US) 2021-12-16 WO disclosed