SCHEMBL2409899

SCHEMBL2409899

COc1cccc(S(=O)(=O)n2cc(CN(CC(C)(C)C)C(=O)O)c(F)c2-c2cccnc2C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.38
CHRM5 P08912 1/20 0.34
NFE2L2 Q16236 1/20 0.34
HTR6 P50406 6/20 0.33
PTGDR2 Q9Y5Y4 3/20 0.33
ELAVL1 Q15717 1/20 0.33
CYP11B1 P15538 1/20 0.32
PLCG1 P19174 1/20 0.32
FGFR4 P22455 1/20 0.32
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP8 P22894 1/20 0.31
MMP13 P45452 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2409876 0.91 HTR6 (0.34) HTR6PTGDR2PLCG1HTR7
SCHEMBL2411542 0.91 MET (0.41) METCHRM5NFE2L2HTR6PTGDR2
SCHEMBL2412057 0.90 PPME1 (0.34) HTR6PTGDR2
SCHEMBL2410603 0.90 HTR6 (0.33) METCHRM5HTR6PTGDR2PLCG1
SCHEMBL2412131 0.89 MET (0.40) METCHRM5NFE2L2HTR6PTGDR2
SCHEMBL4999300 0.89 MET (0.41) METCHRM5NFE2L2HTR6PTGDR2
SCHEMBL2408012 0.87 PTGDR2 (0.31) HTR6PTGDR2PLCG1
SCHEMBL2409898 0.85 MET (0.38) METNFE2L2HTR6ELAVL1PLCG1
SCHEMBL2410118 0.84 PPME1 (0.35) HTR6PTGDR2
SCHEMBL2408074 0.82 HTR6 (0.34) HTR6PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed