SCHEMBL24199813

SCHEMBL24199813

CC(=O)C(C)(C)C(C)(C)N1C(=O)C=CC1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 5/20 0.35
GSK3A P49840 2/20 0.35
GSK3B P49841 2/20 0.35
HSP90AA1 P07900 4/20 0.33
ALDH1A1 P00352 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
HPGD P15428 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
HTT P42858 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
DDAH1 O94760 1/20 0.32
NSD2 O96028 1/20 0.32
G6PD P11413 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
FAAH O00519 1/20 0.32
BLM P54132 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17145360 0.84 MGLL (0.33) MGLLGSK3AGSK3BALDH1A1NPSR1
SCHEMBL23760558 0.81 GSK3A (0.31) MGLLGSK3AGSK3B
SCHEMBL17924887 0.76 MGLL (0.38) MGLLGSK3AGSK3BALDH1A1NPSR1
SCHEMBL18461453 0.75 MGLL (0.41) MGLLGSK3AGSK3BHSP90AA1ALDH1A1
SCHEMBL19882433 0.72 HPGD (0.40) HSP90AA1HPGDPKM
SCHEMBL11509113 0.71 MGLL (0.38) MGLLGSK3AGSK3BHSP90AA1ALDH1A1
SCHEMBL2037967 0.71 MGLL (0.33) MGLLGSK3AGSK3BALDH1A1NPSR1
SCHEMBL18626109 0.71 ALDH1A1 (0.32) MGLLGSK3AGSK3BHSP90AA1ALDH1A1
SCHEMBL8097847 0.70 MGLL (0.41) MGLLGSK3AGSK3BHSP90AA1ALDH1A1
SCHEMBL709031 0.70 MGLL (0.41) MGLLGSK3AGSK3BHSP90AA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558127-B1 TARGETED PYRROLOBENZODIAZEPINE CONJUGATES SEAGEN INC (US) 2022-01-19 EP disclosed